顶体酶抑制剂,acrosin inhibitor
1)acrosin inhibitor顶体酶抑制剂
1.This study is to evaluate if syntheticacrosin inhibitor may affect sperm acrosin.以顶体酶为靶点,第二军医大学药学院药物化学教研室吕加国教授等采用同源模建方法构建人精子顶体酶的三维结构模型,利用InsightII/Bindingsite方法准确定位人精子顶体酶的活性位点,通过柔性分子对接技术建立并合成了一系列顶体酶抑制剂。
2.Objective:To evaluate the inhibitory effect of Nandeshi,anacrosin inhibitor,on human acrosin activity.目的:研究顶体酶抑制剂南德士对人精子顶体酶的抑制作用。
英文短句/例句
1.Sperm Morphological and Functional Modification by Synthetic Acrosin Inhibitor;顶体酶抑制剂对精子形态及功能的影响
2.Characterization of Human Acrosin Active Site and Binding Modes with Its Inhibitors人顶体酶活性腔性质及与抑制剂的结合模式
3.Nandeshi:A Powerful Inhibitor of Human Acrosin Activity南德士抑制人精子顶体酶活性的实验研究
4.Inhibition of Proprotein Convertases by Mung Bean Trypsin Inhibitor;绿豆胰蛋白酶抑制剂对蛋白质前体加工酶的抑制活性
5.Synergistic Effect of Histone Deacetylase Inhibitor SBHA with Proteasome Inhibitors Bortezomib or MG-132 on Breast Cancer Cells;组蛋白去乙酰化酶抑制剂与蛋白酶体抑制剂协同抑制乳腺癌细胞及分子机制研究
6.Effect of the DNA Methyl-transferase Inhibitor on Chromosome of Donor CellsDNA甲基化酶抑制剂对体细胞染色体的影响
7.choline esterase inhibitor胆碱酯酶抑制作用剂
8.nitrate reductase inhibitor硝酸盐还原酶抑制剂
9.soybean trypsin inhibitor大豆胰蛋白酶抑制剂
10.bovine pancreatic trypsin inhibitor牛胰胰蛋白酶抑制剂
11.calpain inhibitor（需）钙蛋白酶抑制剂
12.Inhibiting Effect of Proteasome Inhibitor MG132 on Vascular Stenosis after Balloon Injury & Its Possible Mechanism;蛋白酶体抑制剂MG132抑制球囊损伤后血管狭窄及机制探讨
13.Study of the Effect of Proteasome Inhibitor Bortezomib on Human Pancreatic Cancer Cells;蛋白酶体抑制剂bortezomib在治疗胰腺癌中的实验研究
14.Synthesis of Intermediate of SUN-C8257;糜酶抑制剂SUN-C8257中间体合成方法的研究
15.The Studies on Construction and Application of Screening Model of Proteasome Inhibitor;蛋白酶体抑制剂筛选模型的构建及应用研究
16.Construction of Phage Screening Model for HIV Protease Inhibitor;HIV蛋白酶抑制剂噬菌体筛选模型的构建
17.An Investigation into the Synthesis of C-7 Ingraftation Decorated Steroidal Aromatase Inhibitor;7位接枝修饰的甾体芳香酶抑制剂的合成研究
18.Screening on 171 Natural Natural Products for Proteasomes Inhibitive Activity;171种天然产物蛋白酶体抑制剂活性筛选
相关短句/例句
acrosin inhibitor顶体蛋白酶抑制剂
1.Inhibition effects ofacrosin inhibitor KF 950 on human acrosin;顶体蛋白酶抑制剂KF-950对精子顶体蛋白酶的抑制作用
2.Effects ofacrosin inhibitor 4-guanidinobenzoate on human sperm function;顶体蛋白酶抑制剂4-胍基苯甲酸盐对人精子功能的影响
3)proteasome inhibitor蛋白酶体抑制剂
1.Effect ofproteasome inhibitor and As_2O_3 on expression of survivin mRNA in NB4 cells;蛋白酶体抑制剂联合亚砷酸对NB4细胞survivin基因表达的影响
2.Protective effect ofproteasome inhibitor MG-132 in rats with severe acute pancreatitis and lung injury;蛋白酶体抑制剂MG-132在大鼠重症急性胰腺炎及其肺损伤中的保护作用
3.Toxic effect ofproteasome inhibitor on nigral dopaminergic neuron in mice;蛋白酶体抑制剂对小鼠黑质多巴胺神经元的毒性作用
4)proteasome inhibitors蛋白酶体抑制剂
1.Proteasome andproteasome inhibitors;蛋白酶体与蛋白酶体抑制剂
2.There are many new medicines or new therapies having been developed in recent years,such as thalidomide and its derivant,proteasome inhibitors,arsenic trioxide etc,they are more effective than conventional chemotherapy,such as oral melphalan and prednisone(MP);vincristine,doxorubicin,and dexamethasone(VAD).近年来研制了许多新药或发现了许多药物的新用途,如沙利度胺(thalidom ide)及其衍生物、蛋白酶体抑制剂、砷剂等,与传统的MP、VAD方案相比具有更强的缓解率,给我们的临床工作带来巨大帮助。
3.Furthermore,the effect ofproteasome inhibitors and TAP on particle antigens cross presentation was investigated by FACS analysis.进而,采用流式细胞技术研究了不同蛋白酶体抑制剂以及TAP对噬菌体颗粒抗原交叉呈递的影响。
5)carrier for enzyme inhibitor酶抑制剂载体
6)EI(enzyme-inhibitor complex)酶-抑制剂复合体
延伸阅读
cAMP磷酸二酯酶抑制剂分子式：CAS号：性质：一类能抑制cAMP磷酸二酯酶活性的化合物，是一类具有新机理的强心药。cAMP磷酸二酯酶是在与Ca2+结合的钙调素激活下分解环腺苷酸的酶。cAMP磷酸二酯酶抑制剂能抑制心肌和血管平滑肌细胞内的第三型磷酸二酯酶的活性，使细胞内cAMP含量增加，从而增强心肌收缩，扩张外周血管，改善心力衰竭病人的血流动力学。临床短期使用对急性心力衰竭有明显疗效，但长期使用则引起不良后果。根据对不同亚型的cAMP磷酸二酯酶的亲和力，可分成非选择性抑制剂和选择性抑制剂。
